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Rubio,
B. K.; Robinsion, S. J.; Avalos, C. E.; Valeriote, F. A.; de Voogd, N.
J.; Crews, P. “Revisiting the Sponge Sources, Stereostructure, and
Biological Activity of Cyclocinamide A.” J. Nat. Prod. 2008. (in
press)
Boot,
C. M.; Gassner, N. C.; Compton, J. E.; Tenney, K.; Tamble, C. M.; Lokey, S.;
Holman, T. R.; Crews, P. "Pinpointing Pseurotins from a Marine-Derived Aspergillus
as Tools for Chemical Genetics Using a Synthetic Lethality Yeast
Screen." J. Nat. Prod. 2007, 70, 1671-1675.
Deschamps,
J. D.; Gautschi, J. T.; Whitman, S.; Johnson, T. A.; Gassner, N. C.; Crews,
P.; Holman, T. R. "Discovery of platelet-type 12-human lipoxygenase
selective inhibitors by high-throughput screening of structurally diverse
libraries. Bioorg. Med.
Chem. 2007, 15, 6900-6908.
Boot,
C. M.; Amagata, T.; Tenney, K.; Compton, J. E.; Pietraszkiewicz, H.;
Valeriote, F, A.; Crews, P. "Four Classes of Structurally Unusual
Peptides from two Marine Derived Fungi: Structures and Bioactivities." Tetrahedron
2007, 63, 9903-9914.
Johnson,
T. A.; Tenney, K.; Cichewicz, R. H.; Morinaka, B.; White, K. N.; Amagata, T.; Subramanian,
B.; Media, J,; Mooberry, S. L.; Valeriote, F. A.; Crews, P. "Sponge-Derived
Fijianolides Polyketide Class: Further Evaluation of their Structural and
Cytotoxicity Properties." J. Med. Chem. 2007, 50, 3795-3803.
Hu,
X.; Dang, Y.; Tenney, K.; Crews, P.; Tsai, C. W.; Sixt, D. M.; Cole, P. A.; Liu, J. O. "Regulation
of c-Scr Non-receptor Tyrosine Kinase Activity by Bengamide A through
Inhibition of Metionine Aminopeptidases." Chem. Biol. 2007,
14,
764-774.
Robinson,
S. J.; Tenney, K.; Yee, D.; Martinez, L; Media, J. E.; Valeriote, F. A.; van
Soest, R. W. M.; Crews, P. "Probing the Bioactive Constituents from
Chemotypes of the Sponge Psammocinia aff. bulbosa." J. Nat. Prod. 2007,
70, 1002-1009.
Li,
H.; Amagata, T.; Tenney, K.; Crews, P. "Additional Scalarane
Sesterterpenes from the Sponge Phyllospongia papyracea." J. Nat. Prod.
2007, 70, 802-807.
Rubio,
B. K.; van Soest, R. W. M.; Crews, P. "Extending the Record of
Meroditerpenes from Cacospongia Marine Sponges." J. Nat. Prod. 2007, 70, 628-631.
Piña,
I. C.; White, K. N.; Cabrera, G.; Rivero, E.; Crews, P. "Bromopyrrole
Carboxamide Biosynthetic Products from the Caribbean Sponge Agelas dispar."
J. Nat. Prod. 2007, 70, 613-617.
Gassner,
N. C.; Tamble, C. M.; Bock, J. E.; Cotton, N.; White, K. W.; Tenney, K.; St.
Onge, R. P.; Proctor, M. J.; Giaever, G.; Davis, R. W.; Crews, P.; Holman,
T. R.; Lokey, R. S. "Accelerating the
Discovery of Biologically Active Small Molecules Using a High-Throughput
Yeast Halo Assay." J. Nat. Prod. 2007, 70, 383-390.
Gautschi,
J. T.; Tenney, K.; Compton, J.; Crews, P. "Chemical Investigations of a
Deep Water Marine Derived Fungus: Simple Amino Acid Derivatives from an Arthrinium
sp." Nat. Prod. Comm. 2007, 2, 1-6.
Ralifo,
P.; Sanchez, L.; Gassner, N. C.; Tenney, K.; Lokey, T. S.; Holman, T. R.;
Valeriote, F. A.; Crews, P. "Pyrroloacridine Alkaloids from Plakortis
quasiamphiaster: Structures and Bioactivity." J. Nat. Prod. 2007, 70, 95-99.
Wegerski,
C. J.; Hammond, J.; Tenney, K.; Matainaho, T.; Crews, P. "A
Serendipitous Discovery of Isomotuporin-Containing Sponge Populations of
Theonella swinhoei." J. Nat. Prod.
2007, 70, 89-94.
Ralifo,
P.; Tenney, K.; Valeriote, F. A.; Crews, P. "A Distinctive Structural
Twist in the Aminoimidazole Alkaloids from a Calcareous Marine Sponge:
Isolation and Characterization of Leucosolenamenes A and B." J. Nat.
Prod. 2007, 70, 33-38.
Amagata,
T.; Morinaka, B. I.; Amagata, A.; Tenney, K.; Valeriote, F. A.; Lobkobsky,
E.; Clardy, J.; Crews, P. "A Chemical Study of Cyclic Depsipeptides
Produced by a Sponge-Derived fungus." J. Nat. Prod. 2006,
69,
1560-1565.
Wegerski,
C. J.; Sonnenschein, R. N.; Cabriales, F.; Valeriote, F. A.; Matainago, T.;
Crews. P. "Stereochemical Challenges in Characterizing Nitrogenous
Spiro-Axane Sesquiterpenes fromthe Indo-Pacific Sponges Amorphinopsis and Axinyssa."
Tetrahedron 2006, 62, 10393-10399.
Sonnenschein,
R. N.; Johnson, T. A.; Tenney, K.; Valeriote, F. A.; Crews, P. "A
Reassignment of (-)-Mycothiazole and the Isolation of a Related Diol." J.
Nat. Prod. 2006, 69, 145-147
Subramanian,
B.; Nakeff, A.; Tenney, K.; Crews, P.; Gunatilaka, L.; Valeriote, F. "A
New Paradigm for the Development of Anticancer Agents from Natural
Products." Journal of Experimental Therapeutics and Oncology.
2006, 5, 195-204.
Boot, C.
M.; Tenney, K.; Valeriote, F. A.; Crews, P. "Highly N-methylated LInear
Peptides Produced by an Atypical Sponge-Derived Acremonium sp." J.
Nat. Prod. 2006, 69, 83-92.
Christian,
O. E.; Compton, J.; Christian, K. R.; Mooberry, S. L.; Valeriote, F. A.;
Crews, P. "Using Jasplakinolide to Turn on Pathways that Enable the
Isolation of New Chaetoglobosins from Phomopsis asparagi." J. Nat.
Prod. 2005, 68, 1592-1597.
Segraves, N. L.; Crews, P.
"Invesigation of Brominated Tryptophan Alkaloids from Two Thorectidae
Sponges: Thorectandra and Smenospongia." J. Nat. Prod. 2005,
68,
1484-1488.
Cichewicz,
R. H.; Clifford, L. J.; Lassesn, P. R.; Cao, X.; Freedman, T. B.; Nafie, L.
A.; Deschamps, J. D.; Kenyon, V. A.; Flanary, J. R.; Holman, T. R.; Crews,
P. "Stereochemical Determination and Bioactivity Assessment of (S)-(+)-Curcuphenol
Dimers Isolated from the Marine Sponge Didiscus aceratus and Synthesized
through Laccase Biocatalysis." Bio. Med. Chem. 2005,
13,
5600-5612.
Segraves, N. L.; Crews, P.
"A Madagascar Sponge Batzella sp. as a Source of
Alkylated Iminosugars." J. Nat. Prod. 2005,
68, 118-121.
Ralifo.
P; Crews, P. "A New Structural Theme in the Imidazole Containing
Alkaloids from a Calcareous Leucetta Sponge". J.
Org. Chem. 2004, 69, 9025-9029.
Cichewicz, R. H.; Kenyon,
V. A.; Whitman, S.; Morales, N. M.; Arguello, J. F.; Holman, T. R.; Crews,
P. "Redox Inactivation of Human 15-Lipoxygenase by Marine-Derived
Meroditerpenes and Synthetic Chromanes:
Archetypes for a Unique Class of Selective and Recyclable
Inhibitors". J. Am. Chem. Soc. 2004, 126,
14910-14920.
Wegerski,
C. J.; France, D.; Cornell-Kennon, S.; Crews, P. "Using a Kinase Screen
to Investigate the Constituents of the Sponge Stelleta clavosa
Obtained from Diverse Habitats". Bioorg. Med. Chem. 2004, 12, 5631-5637.
Segraves, E. N.; Shah, R.
R.; Segraves, N. L.; Johnson, T. A.; Whitman, S.; Sui, J. K.; Kenyon, V. A.;
Cichewicz, R. H.; Crews, P.; Holman, T. R. "Probing the Activity
Differences of Simple and Complex Brominated Aryl Compounds against
15-Soybean, 15-Human and 12-Human Lipoxygenases". J. Med. Chem. 2004, 47, 4060-4065.
Gautschi, J. T.; Whitman, S.;
Holman, T. R.; Crews, P. "An Analysis of Phakellin and Oroidin
Structures Stimulated by Further Study of an Agelas Sponge". J.
Nat. Prod. 2004, 67, 1256-1261.
Vilozny, B.; Amagata, T.;
Mooberry, S. L.; Crews, P. "A New Dimension to the Biosynthetic
Products Isolated from the Sponge Negombata magnifica". J.
Nat. Prod. 2004, 67, 1055-1057.
Cichewicz, R. H.; Valeriote,
F. A.; Crews, P. "Psymberin, A Potent Sponge- Derived
Cytotoxin from Psammocinia Distantly Related to the Pederin Family". Org.
Lett. 2004, 6, 1951-1954.
Segraves, N. L.; Robinson,
S. J.; Garcia, D.; Said, S. A.; Fu, X.; Schmitz, F. J.; Petraszkiewicz, H.;
Valeriote, F. A.; Crews, P. "Comparison of Fascaplysin and Related
Alkaloids – A Study of Structures, Cytotoxicities, and Sources". J.
Nat. Prod. 2004, 67, 783-792.
Gautschi, J. T.; Amagata,
T.; Amagata, A.; Valeriote, F. A.; Mooberry, S. L.; Crews, P. "Expanding
the Strategies in Natural Product Studies of Marine-Derived Fungi: A
Chemical Investigation of Penicillium Obtained from Deep Water
Sediment". J. Nat. Prod. 2004, 67, 362-367.
Sonnenschein, R. N.; Farias,
J. J.; Tenney, K.; Mooberry, S. L.; Lobkovsky, E.; Clardy, J.; Crews, P.
"A Further Study of the Cytotoxic Constituents of a Milnamide Producing
Sponge". Org. Lett. 2004, 6, 779-782.
Lepourcelet, M.; Chen,
Y.-N. P.; France, D. S.; Wang, H.; Crews, P.; Petersen, F.; Bruseo, C.;
Wood, A. W.; Shivdasani, R. "A. Small-Molecule Antagonists of the
Oncogenic Tcf/b-Catenin Protein Complex". Cancer Cell 2004, 5, 91-102.
Crews, P.; Gerwick, W. H.;
Schmitz, F. J.; France, D.; Bair, K. W.; Wright, A. E.; Hallock, Y. "Molecular
Approaches to Discover Marine Natural Product Anticancer Leads – An Update
from a Drug Discovery Group Collaboration". Pharm. Biol. 2003, 41, 39-52.
Amagata, T.; Amagata, A.;
Tenney, K.; Valeriote, F. A.; Lobkovsky, E.; Clardy, J.; Crews, P. "Unusual
C25 Steroids Produced by a Sponge-Derived Penicillium citrinum".
Org. Lett. 2003, 5, 4393-4396.
Amagata, T.; Rath, C.; Rigot, J.
F.; Tarlov, N.; Tenney, K.; Valeriote, F. A.; Crews, P. "Structures and
Cytotoxic Properties of Trichoverroids and their Macrolide Analogues
Produced by Saltwater Culture of Myrothecium verrucaria". J. Med.
Chem. 2003, 46, 4342-4350.
Edrada, R. A.; Stessman, C. C.;
Crews, P. "Uniquely Modified Imidazole Alkaloids from a Calcareous Leucetta
Sponge". J. Nat. Prod. 2003, 66, 939-942.
Wenzel, P. J.; Crews, P. "Probing
Biotransformation Relationships Among Pyridoacridines by Focusing on
Oxygenated Analogs". J. Nat. Prod. 2003, 66,
873-875.
Piña, I. C.; Gautschi, J. T.;
Wang, G.-Y.-S.; Sanders, M. L.; Schmitz, F. J.; France, D.; Cornell-Kennon,
S.; Sambucetti, L. C.; Remiszewski, S. W.; Bair, K. W.; Crews, P. "Psammaplins
from the Sponge Psuedoceratina purpurea: Inhibition of Both Histone
Deacetylase and DNA Methyltransferase". J. Org. Chem. 2003, 68, 3866-3873.
Segraves, N. L.; Lopez, S.;
Johnson, T. A.; Said, S. A.; Fu, X.; Schmitz, F. J.; Pietraszkiewicz, H.;
Valeriote, F. A.; Crews, P. "Structures and Cytotoxicities of
Fascaplysin and Related Alkaloids from Two Marine Phyla - Fascaplysinopsis
Sponges and Didemnum Tunicates". Tetrahedron Lett. 2003, 44, 3471-3475.
Amagata, T.; Whitman, S.;
Johnson, T. A.; Stessman, C. C.; Loo, C.; Lobkovsky, E.; Clardy, J.; Crews,
P.; Holman, T. R. "Explored Sponge-Derived Terpenoids for their Potency
and Selectivity Against 12-Human, 15-Human, and 15-Soybean Lipoxygenases".
J. Nat. Prod. 2003, 66, 230-235.
Crews, P.; Clark, D. P.; Tenney,
K. "Variation in the Alkaloids Among Indo-Pacific Leucetta
Sponges". J. Nat. Prod. 2003, 66, 177-182.
Piña, I. C.; Sanders, M. L.; Crews, P. "Puupehenone Congeners from an Indo- Pacific Hyrtios Sponge". J. Nat. Prod. 2003, 66, 2-6.